[1]魏士雄 孙赫.过氧化物酶体增殖物激活受体激动剂在心肌梗死中的作用机制研究进展[J].心血管病学进展,2021,(12):1110-1113.[doi:10.16806/j.cnki.issn.1004-3934.2021.12.013]
 WEI Shixiong,SUN He.Action Mechanism of Peroxisome Proliferator-activated Receptor Agonist in Myocardial Infarction[J].Advances in Cardiovascular Diseases,2021,(12):1110-1113.[doi:10.16806/j.cnki.issn.1004-3934.2021.12.013]
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过氧化物酶体增殖物激活受体激动剂在心肌梗死中的作用机制研究进展()
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《心血管病学进展》[ISSN:51-1187/R/CN:1004-3934]

卷:
期数:
2021年12期
页码:
1110-1113
栏目:
综述
出版日期:
2021-12-25

文章信息/Info

Title:
Action Mechanism of Peroxisome Proliferator-activated Receptor Agonist in Myocardial Infarction
作者:
魏士雄 孙赫
(吉林大学白求恩第一医院胸心外科,吉林 长春 130000)
Author(s):
WEI ShixiongSUN He
(Department of Cardiothoracic Surgery,The First Bethune Hospital of Jilin University,Changchun 130000,Jilin,China)
关键词:
过氧化物酶体增殖物激活受体心肌梗死血管生成心肌细胞
Keywords:
Peroxisome proliferator-activated receptorMyocardial infarctionAngiogenesisCardiomyocytes
DOI:
10.16806/j.cnki.issn.1004-3934.2021.12.013
摘要:
过氧化物酶体增殖物激活受体(PPARs)属于核激素受体家族的一员,是一类由配体激活的转录因子,包括PPARα、PPARβ/δ和PPARγ三种亚型。PPARs已被证实具有调节血糖水平、脂质稳态、炎症发展和机体发育在内的多种功能,且能够在不同的组织和细胞中特异性表达。既往研究已明确PPARs激动剂在治疗糖尿病和高脂血症中的重大作用,近来PPARs配体作为心血管疾病治疗靶点的潜在价值也引起了学者们的广泛关注。现综述PPARs激动剂对心肌梗死情况影响的基础和临床研究进展,并对未来进一步的深入研究方向提出设想。
Abstract:
Peroxisome proliferator-activated receptors(PPARs) belong to nuclear hormone receptor family. They are ligand-activated transcription factors and exist in three isoforms,PPARα,PPARβ/δ,and PPARγ. PPARs regulate a variety of functions,including glucose and lipid homeostasis,inflammation,and body development. They exhibit tissue and cell type-specific expression patterns and functions. Besides the established notion of the therapeutic potential of PPAR agonists for the treatment of glucose and lipid disorders,more recent data proposed specific PPAR s ligands as potential therapies for cardiovascular diseases. Here we review the basic and clinical research results of the effects of PPARs agonists on myocardial infarction ,and proposes ideas for further in-depth research in the future.

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备注/Memo

备注/Memo:
基金项目:军委后勤保障部卫生局面上项目(16BJZ28)
通信作者:孙赫,E-mail:773691039@qq.com
收稿日期:2021-08-04
更新日期/Last Update: 2022-01-07