[1]孟凡华 付真彦.一种新型的治疗血脂异常的干扰RNA药物Inclisiran[J].心血管病学进展,2021,(2):167.[doi:10.16806/j.cnki.issn.1004-3934.2021.02.018]
 MENG Fanhua,FU Zhenyan.Inclisiran, A New Small Interfering RNA Drug for the Treatment of Dyslipidemia[J].Advances in Cardiovascular Diseases,2021,(2):167.[doi:10.16806/j.cnki.issn.1004-3934.2021.02.018]
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一种新型的治疗血脂异常的干扰RNA药物Inclisiran()
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《心血管病学进展》[ISSN:51-1187/R/CN:1004-3934]

卷:
期数:
2021年2期
页码:
167
栏目:
综述
出版日期:
2021-02-25

文章信息/Info

Title:
Inclisiran, A New Small Interfering RNA Drug for the Treatment of Dyslipidemia
作者:
孟凡华 付真彦
(新疆医科大学第一附属医院心脏中心,新疆 乌鲁木齐 830000)
Author(s):
MENG Fanhua FU Zhenyan
 (The First Affiliated HospitalXinjiang Medical University,Urumqi 830000,Xinjiang,China)
关键词:
InclisiranRNA血脂异常前蛋白转化酶枯草溶菌素9
Keywords:
InclisiranRNADyslipidemiaPCSK9
DOI:
10.16806/j.cnki.issn.1004-3934.2021.02.018
摘要:
Inclisiran是第一个用于降血脂的干扰RNA药物,它能特异性抑制前蛋白转化酶枯草溶菌素9的合成,从而降低低密度脂蛋白胆固醇,具有良好的有效性和安全性。现综述目前国内外关于Inclisiran作为降脂药物预防心血管疾病的作用机制、有效性和安全性。
Abstract:
Inclisiran is the first small interfering RNA drug for lipid lowering,which can specifically inhibit the synthesis of the proprotein convertase subtilisin/kexin type 9,thus lowering LDL cholesterol,with good efficacy and safety. This review summarizes the mechanism,effectiveness and safety of Inclisiran as a lipid-lowering drug to prevent cardiovascular diseases

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更新日期/Last Update: 2021-06-16