[1]邓皓月,综述,陈明,等.升高高密度脂蛋白胆固醇药物的研究进展[J].心血管病学进展,2016,(3):258-262.[doi:10.16806/j.cnki.issn.1004-3934.2016.03.011]
 DENG Haoyue,CHEN Ming.Advances in Elevating High-density Lipoprotein Cholesterol Drugs[J].Advances in Cardiovascular Diseases,2016,(3):258-262.[doi:10.16806/j.cnki.issn.1004-3934.2016.03.011]
点击复制

升高高密度脂蛋白胆固醇药物的研究进展()
分享到:

《心血管病学进展》[ISSN:51-1187/R/CN:1004-3934]

卷:
期数:
2016年3期
页码:
258-262
栏目:
综述
出版日期:
2016-06-20

文章信息/Info

Title:
Advances in Elevating High-density Lipoprotein Cholesterol Drugs
作者:
邓皓月综述陈明审校
重庆医科大学附属第一医院心内科,重庆 400016
Author(s):
DENG HaoyueCHEN Ming
Department of Cardiology,The First Affiliated Hospital of Chongqing Medical University,Chongqing 400016,China
关键词:
高密度脂蛋白胆固醇 胆固醇逆向转运 烟酸 胆固醇酯转移蛋白抑制剂
Keywords:
High-density lipoprotein cholesterol Reverse cholesterol transport Nicotinic acid Cholesterol ester transfer protein inhibitor
分类号:
R972+.6
DOI:
10.16806/j.cnki.issn.1004-3934.2016.03.011
文献标志码:
A
摘要:
冠心病严重危害到人们的生命及身体健康,而大量流行病学研究表明高密度脂蛋白胆固醇水平与患冠心病的风险呈负相关,故升高高密度脂蛋白胆固醇成为治疗冠心病的又一热点,目前能有效升高高密度脂蛋白胆固醇而又带来明确心血管获益的药物尚少,大多处于研究阶段,且仍具有临床争议,现在讲述可升高高密度脂蛋白胆固醇的传统调脂药物以及特异性升高高密度脂蛋白胆固醇的药物的最新研究进展。
Abstract:
Coronary heart disease is a serious threat to people's life and health. A large number of epidemiological studies have indicated that high-density lipoprotein cholesterol is negatively associated with the risk of coronary heart disease. The increase of high-density lipoprotein cholesterol has become a hot issues for the treatment of coronary heart disease, which can effectively increase the high-density lipoprotein cholesterol. Presently drugs that can effectively increase high-density lipoprotein cholesterol and have clear cardiovascular benefits are mostly in the research stage, and are still controversial. This paper describes the latest research progress of the drug that can specifically increase the cholesterol of high-density lipoprotein cholesterol and the traditional lipid regulating drugs.

参考文献/References:

[1] Chyu KY, Shah PK. HDL/ApoA-1 infusion and ApoA-1 gene therapy in atherosclerosis[J]. Front Pharmacol,2015,6:187.
[2] Kingwell BA, Chapman MJ, Kontush A,et al. HDL-targeted therapies:progress, failures and future[J]. Nat Rev Drug Discov,2014,13(6):445-464.
[3] Wang M,Briggs MR. HDL:the metabolism, function,and therapeutic importance[J]. Chem Rev,2004,104(1):119-137.
[4] Jacobson TA, Ito MK,Maki KC,et al. National Lipid Association recommendations for patient-centered management of dyslipidemia:part 1—executive summary[J].J Clin Lipidol,2014,8(5):473-488.
[5] Goyal P, Igel LI, LaScalea K,et al. Cardiometabolic impact of non-statin lipid low-ering therapies[J]. Curr Atheroscler Rep,2014,16:390.
[6] Sando KR,Michelle Knight P.Nonstatin therapies for management of dyslipidemia: a review[J]. Clin Ther,2015,37(10):2153-2179.
[7] Gomaraschi M, Adorni MP, Banach M, et al. Effects of established hypolipidemic drugs on HDL concentration, subclass distribution,and function[J].Handb Exp Pharmacol,2015,224:593-615.
[8] Rubins HB,Robins SJ,Collins D,et al.Gemfibrozil for the secondary prevention of coronary heart disease in men with low levels of high-density lipoprotein cholesterol.Veterans Affairs High-density Lipoprotein Cholesterol Intervention Trial Study Group[J].N Engl J Med,1999,341(6):410-418.
[9] Ginsberg HN. The ACCORD(Action to Control Cardiovascular Risk in Diabetes)Lipid Trial: What we learn from subgroup analyses[J]. Diabetes Care,2011,34(Suppl 2):S107-108.
[10] Yadav R,Liu Y,Kwok S,et al.Effect of extended-release niacin on high-density lipoprotein(HDL)functionality, lipoprotein metabolism, and mediators of vascular inflammation in statin-treated patients[J]. J Am Heart Assoc,2015,4(9):e001508.
[11] Mani P,Rohatgi A.Niacintherapy, HDL cholesterol, and cardiovascular disease: is the HDL hypothesis defunct? [J]. Curr Atheroscler Rep,2015,17(8):521.
[12] Zeman M, Vecka M, Perlík F, et al. Niacin in the treatment of hyperlipidemias in light of new clinical trials:has niacin lost its place?[J]. Med Sci Monit,2015,21:2156-2162.
[13] Keene D, Price C, Shun-Shin MJ, et al.Effect on cardiovascular risk of high density lipoprotein targeted drug treatments niacin,fibrates,and CETP inhibitors: meta-analysis of randomized controlled trials including 117 411 patients[J]. BMJ, 2014,349:g4379.
[14] Krause BR, Remaley AT. Reconstituted HDL for the acute treatment of acute coronary syndrome[J].Curr Opin Lipidol,2013,24(6):480-486.
[15] Hafiane A, Kellett S, Genest J. Treatment options for low high-density lipoproteins[J]. Curr Opin Endocrinol Diabetes Obes,2014,21(2):134-139.
[16] Joy TR. Novel HDL-based therapeutic agents[J]. Pharmacol Ther,2012,135(1):18-30.
[17] Bishop Bryan M. Systematic review of CETP inhibitors for increasing high-density lipoprotein cholesterol: where do these agents stand in the approval process?[J]. Am J Ther,2015,22(2):147-158.
[18] Hovingh GK, Kastelein JJ, van Deventer SJ, et al. Cholesterol ester transfer protein inhibition by TA-8995 in patients with mild dyslipidaemia(TULIP):a randomised, double-blind, placebo-controlled phase 2 trial[J]. Lancet,2015,386(9992): 452-460.
[19] Ford J,Lawson M,Fowler D,et al.Tolerability,pharmacokinetics and pharmacodynamics of TA-8995, a selective cholesteryl ester transfer protein(CETP)inhibitor, in healthy subjects[J]. Br J Clin Pharmacol,2014,78(3):498-508.
[20] Rittershaus CW,Miller DP,Thomas LJ, et al. Vaccine-induced antibodies inhibit CETP activity in vivo and reduce aortic:lesions in a rabbit model of atherosclerosis[J]. Arterioscler Thromb Vasc Biol,2000,20(9):2106-2112.
[21] Salazar-González JA,Rosales-Mendoza S. A perspective for atherosclerosis vaccination:is there a place for plant-based vaccines?[J]. Vaccine,2013,31(10):1364-1349.
[22] Liaw YW, Lin CY, Lai YS, et al.A vaccine targeted at CETP alleviates high fat and high cholesterol diet-induced atherosclerosis and non-alcoholic steatohepatitis in rabbit[J]. PLoS One,2014,9(12):e111529.
[23] Scharnagl H,Heuschneider C,Sailer S,et al. Decreased cholesterol efflux capacity in patients with low cholesteryl ester transfer protein plasma levels[J]. Eur J Clin Invest,2014,44(4):395-401.
[24] Mousa SS, Block RC, Mousa SA. High density lipoprotein(HDL)modulation targets[J]. Drugs Future,2010,35(1):33-39.
[25] Peng D,Hiipakka RA,Dai Q, et al.Antiatherosclerotic effects of a novel synthetic tissue-selective steroidal liver X receptor agonist in low-density lipoprotein receptor-deficient mice[J]. J Pharmacol Exp Ther,2008,327(2):332-342.
[26] Pfeifer T, Buchebner M, Chandak PG, et al.Synthetic LXR agonist suppresses endogenous cholesterol biosynthesis and efficiently lowers plasma cholesterol[J]. Curr Pharm Biotechnol,2011,12(2):285-292.
[27] Fievet C,Staels B.Liver X receptor modulators:effects on lipid metabolism and potential use in the treatment of atherosclerosis[J].Biochem Pharmacol,2009,77(8): 1316-1327.
[28] Omidi A,Ansarinik H,Ghazaghi M. Prosopis farcta beans increase HDL cholesterol and decrease LDL cholesterol in ostriches( Struthio camelus )[J]. Trop Anim Health Prod,2013,45(2):431-434.
[29] McEneny J,Wade L,Young IS,et al.Lycopene intervention reduces inflammation and improves HDL functionality in moderately overweight middle-aged individuals[J]. J Nutr Biochem,2013,24(1):163-168.
[30] van de Woestijne AP,van der Graaf Y,Liem AH,et al.Low high-density lipoprotein cholesterol is not a risk factor for recurrent vascular events in patients with vascular disease on intensive lipid-lowering medication[J]. J Am Coll Cardiol,2013,62(20):1834-1841.
[31] Rohatgi A. High-density lipoprotein function measurement in human studies: focus on cholesterol efflux capacity[J]. Prog Cardiovasc Dis,2015,58(1):32-40.

相似文献/References:

[1]刘力黎 陈诚 张丽敏.血脂水平与心房颤动相关性研究进展[J].心血管病学进展,2021,(6):539.[doi:10.16806/j.cnki.issn.1004-3934.2021.06.015]
 LIU Lili,CHEN Cheng,ZHANG Limin.Serum Lipid Level and Atrial Fibrillation[J].Advances in Cardiovascular Diseases,2021,(3):539.[doi:10.16806/j.cnki.issn.1004-3934.2021.06.015]
[2]陈旭东 黄春霞 高奋.高密度脂蛋白胆固醇与心房颤动发生的研究进展[J].心血管病学进展,2023,(10):930.[doi:10.16806/j.cnki.issn.1004-3934.2023.10.015]
 CHEN XudongHUANG ChunxiaGAO Fen.High-Density Lipoprotein Cholesterol and Atrial Fibrillation[J].Advances in Cardiovascular Diseases,2023,(3):930.[doi:10.16806/j.cnki.issn.1004-3934.2023.10.015]

备注/Memo

备注/Memo:
作者简介:邓皓月(1991—),住院医师,在职硕士,主要从事冠状动脉粥样硬化性心脏病研究。Email:1067192362@qq.com 通信作者:陈明(1962—),教授,主任医师,博士,主要从事高血压研究。Email: chenmingcq@126.com
更新日期/Last Update: 2016-05-25